BDBM709474 6-(1-(1-(9-acryloyl-3-oxa- 7,9- diazabicyclo[3.3.1]nonane- 7-carbonyl)piperidin-4- yl)-1H-pyrazol-4-yl)-4- methoxypyrazolo[1,5- a]pyridine-3-carbonitrile::US12180207, Example 3

SMILES C=CC(=O)N1C2COCC1CN(C(=O)N1CCC(n3cc(-c4cc(OC)c5c(C#N)cnn5c4)cn3)CC1)C2

InChI Key

Data  5 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 709474   

TargetFibroblast growth factor receptor 1(Human)
Array Biopharma

US Patent
LigandPNGBDBM709474(6-(1-(1-(9-acryloyl-3-oxa- 7,9- diazabicyclo[3.3.1...)
Affinity DataIC50: 44nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 3(Human)
Array Biopharma

US Patent
LigandPNGBDBM709474(6-(1-(1-(9-acryloyl-3-oxa- 7,9- diazabicyclo[3.3.1...)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 1(Human)
Array Biopharma

US Patent
LigandPNGBDBM709474(6-(1-(1-(9-acryloyl-3-oxa- 7,9- diazabicyclo[3.3.1...)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 2(Human)
Array Biopharma

US Patent
LigandPNGBDBM709474(6-(1-(1-(9-acryloyl-3-oxa- 7,9- diazabicyclo[3.3.1...)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent

TargetFibroblast growth factor receptor 3(Human)
Array Biopharma

US Patent
LigandPNGBDBM709474(6-(1-(1-(9-acryloyl-3-oxa- 7,9- diazabicyclo[3.3.1...)
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
5/12/2025
Entry Details
Go to US Patent