BDBM684597 1-(3'-(5-(4-(tert- butyl)piperazin-1- yl)-6-methoxypyri- din-3-yl)-3-chloro- 5'-fluoro-2'-hydroxy- [1,1'-biphenyl]-4- yl)-3-methyl-1,3- dihydro-2H-imid- azol-2-one::US20240226096, Example I-15

SMILES COc1ncc(cc1N1CCN(CC1)C(C)(C)C)-c1cc(F)cc(c1O)-c1ccc(c(Cl)c1)-n1ccn(C)c1=O

InChI Key InChIKey=BPGDMNMQPOTZCY-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 684597   

TargetBromodomain-containing protein 4 [368-440](Human)
Poseidon Innovation 1

US Patent
LigandPNGBDBM684597(US20240226096, Example I-15 | 1-(3'-(5-(4-(tert- b...)
Affinity DataIC50: 0.152nMAssay Description:3x Complete Substrate plus Inhibitor Solution in Assay Medium (Opti-MEM I Reduced Serum Medium, no phenol red, and no serum) was prepared just before...More data for this Ligand-Target Pair
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US Patent