BDBM681891 US20240199649, Compound 754

SMILES Cc1nc2ccc(nc2n1CC(F)(F)F)-c1ccn2nc(N[C@H]3CC[C@](C)(O)CC3)nc(N)c12

InChI Key InChIKey=LZZMPPFSEPQRPF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 681891   

TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Human)
Biosplice Therapeutics

US Patent
LigandPNGBDBM681891(US20240199649, Compound 754)
Affinity DataIC50: 0.5nMAssay Description:The DYRK1A kinase assay was run using the Ser/Thr 18 peptide Z-lyte assay kit according to manufacturer's instructions (Life Technologies a Division ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2024
Entry Details
Go to US Patent