BDBM675063 1-(5-(4-amino-7-(piperidin-4- yl)-7H-pyrrolo[2,3-d]pyr- imidin-5-yl)imidazo[1,2-a]- pyridin-8-yl)-3-(4-((4-methyl- piperazin-1-yl)methyl)-3- (trifluoromethyl)phenyl)urea::US20240158394, Compound I-133

SMILES CN1CCN(Cc2ccc(NC(=O)Nc3ccc(-c4cn(C5CCNCC5)c5ncnc(N)c45)n4ccnc34)cc2C(F)(F)F)CC1

InChI Key InChIKey=HRJQQAILMKESKU-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 675063   

TargetSerine/threonine-protein kinase Nek7(Human)
Halia Therapeutics

US Patent
LigandPNGBDBM675063(1-(5-(4-amino-7-(piperidin-4- yl)-7H-pyrrolo[2,3-d...)
Affinity DataIC50: 200nMAssay Description:Casein substrate (from bovine milk, hydrolyzed and partially dephosphorylated mixture of α, β and κ caseins, obtained from Sigma Aldri...More data for this Ligand-Target Pair
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US Patent