BDBM621052 US20230303556, Compound Formula (C)
SMILES C[C@H]1CN(C[C@@H](C)N1)c1cc(cc2n(ncc12)-c1nnc(s1)C(F)F)S(=O)(=O)NC1(C)CC1
InChI Key InChIKey=AQOUTSJIZZVANZ-UHFFFAOYSA-N
Data 1 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 621052
Affinity DataEC50: 15nMAssay Description:PARG enzyme was incubated with compound or vehicle (DMSO) and the biotinylated-PARylated PARP-1 substrate in a microtiter plate. After adding detecti...More data for this Ligand-Target Pair