BDBM615667 (1R,5S,6r)-N-(propan-2-yl)-3-[5-(propan-2-yl)-1H-pyrazole-3-carbonyl]-3-azabicyclo[3.1.0]hexane-6-carboxamide::US20230271952, Example 136

SMILES CC(C)NC(=O)[C@@H]1[C@H]2CN(C[C@@H]12)C(=O)c1cc([nH]n1)C(C)C

InChI Key InChIKey=IXZBELFRWCXTJD-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 615667   

TargetLysine-specific demethylase 5A(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM615667((1R,5S,6r)-N-(propan-2-yl)-3-[5-(propan-2-yl)-1H-p...)
Affinity DataIC50: 50nMAssay Description:Using 384-well white Greiner784075 (Greiner), representative compounds were characterized for their inhibition of KDM5A using HTRF technology (Cisbio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2023
Entry Details
Go to US Patent