BDBM615640 (1-isopropyl-1H-imidazol-4-yl)[(1R,5S,6r)-6-([1,2,3]triazolo[1,5-a]pyridin-3-yl)-3-azabicyclo[3.1.0]hex-3-yl]methanone::US20230271952, Example 62

SMILES CC(C)n1cnc(c1)C(=O)N1C[C@H]2[C@@H](C1)[C@@H]2c1nnn2ccccc12

InChI Key InChIKey=RIQDTFFFDKPBAU-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 615640   

TargetLysine-specific demethylase 5A(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM615640((1-isopropyl-1H-imidazol-4-yl)[(1R,5S,6r)-6-([1,2,...)
Affinity DataIC50: 10nMAssay Description:Using 384-well white Greiner784075 (Greiner), representative compounds were characterized for their inhibition of KDM5A using HTRF technology (Cisbio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2023
Entry Details
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