BDBM615634 US20230271952, Example 40::{(1R,5S,6r)-6-[5-(difluoromethyl)-5-methyl-4,5-dihydro-1,2-oxazol-3-yl]-3-azabicyclo[3.1.0]hex-3-yl}(1-isopropyl-1H-imidazol-4-yl)methanone

SMILES CC(C)n1cnc(c1)C(=O)N1C[C@H]2[C@@H](C1)[C@@H]2C1=NOC(C)(C1)C(F)F

InChI Key InChIKey=MHYJPOVWHJXQEI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 615634   

TargetLysine-specific demethylase 5A(Human)
Ono Pharmaceutical

US Patent
LigandPNGBDBM615634({(1R,5S,6r)-6-[5-(difluoromethyl)-5-methyl-4,5-dih...)
Affinity DataIC50: 200nMAssay Description:Using 384-well white Greiner784075 (Greiner), representative compounds were characterized for their inhibition of KDM5A using HTRF technology (Cisbio...More data for this Ligand-Target Pair
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Date in BDB:
10/16/2023
Entry Details
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