BDBM608342 US11691981, Compound 79

SMILES CC1(C)OC(=O)c2ccc(Nc3cc(Oc4cn(nc4C4CCOCC4)C4CC4)ccn3)cc12

InChI Key InChIKey=QZXHEAXOKDPRNW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 608342   

TargetTGF-beta receptor type-1(Human)
Inventisbio

US Patent
LigandPNGBDBM608342(US11691981, Compound 79)
Affinity DataIC50: 29nMAssay Description:TGFβR1 kinase assay was performed according to the instruction manual of the ADP-Glo™ Kinase Assay kit provided by Promega. Prepare 1× Kina...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2023
Entry Details
Go to US Patent