BDBM605039 US11667643, Compound I-73

SMILES Clc1nc2C(CCc3ccccc3-n2c1Cl)NC(=O)c1ncn(Cc2c(Cl)cccc2Cl)n1

InChI Key InChIKey=FSFFJENCZPESBL-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 605039   

TargetReceptor-interacting serine/threonine-protein kinase 1(Human)
Rigel Pharmaceuticals

US Patent
LigandPNGBDBM605039(US11667643, Compound I-73)
Affinity DataIC50: 92.4nMAssay Description:ADP-Glo (Promega, Madison, Wis., USA) reagents were thawed at ambient temperature. Kinase Detection Reagent was prepared by mixing kinase detection b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/9/2023
Entry Details
Go to US Patent