BDBM579121 US11479560, Title DM-68::US11479560, Title ww4-105

SMILES Cc1ccc(CC(CO)n2c3ccccc3n(Cc3nc4ccccc4o3)c2=N)cc1

InChI Key InChIKey=DURUHVZIDVXKAG-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 579121   

TargetOrexin receptor type 2(Human)
University of Texas System

US Patent
LigandPNGBDBM579121(US11479560, Title ww4-105 | US11479560, Title DM-6...)
Affinity DataEC50: >1.00E+3nMAssay Description:HEK293 cells stably expressing OX2R are transfected with Gq alpha construct (6.4 ug per 10 cm dish) using Lipofectamine 3000 (ThermoFisher). 24 hours...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
Go to US Patent

TargetOrexin receptor type 2(Human)
University of Texas System

US Patent
LigandPNGBDBM579121(US11479560, Title ww4-105 | US11479560, Title DM-6...)
Affinity DataEC50:  5.00E+3nMAssay Description:HEK293 cells stably expressing OX2R are transfected with Gq alpha construct (6.4 ug per 10 cm dish) using Lipofectamine 3000 (ThermoFisher). 24 hours...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
Go to US Patent