BDBM564302 US11414384, Example 102 Isomer 4
SMILES C[C@@H](CN[C@@H](C(=O)c1cnn2cc(ccc12)-c1cnn(C)c1)c1ccccc1)c1ccc(cc1)C#N
InChI Key InChIKey=OJALLZBPDOMARU-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 564302
TargetHistone acetyltransferase p300 [1287-1666]/Histone acetyltransferase type B catalytic subunit(Human)
Constellation Pharmaceuticals
US Patent
Constellation Pharmaceuticals
US Patent
Affinity DataIC50: 9.36nMAssay Description:The p300 HAT domain (residues 1287-1666) was expressed and purified with an N-terminal His tag from Escherichia coli cells. The expressed protein was...More data for this Ligand-Target Pair