BDBM538081 4-(4-fluoro-3-(1-isopropyl-4-oxido-1,4-azaphosphinan-4-yl)benzyl)phthalazin-1(2H)-one::US11248013, Example 42
SMILES CC(C)N1CCP(=O)(CC1)c1cc(Cc2n[nH]c(=O)c3ccccc23)ccc1F
InChI Key InChIKey=BGPIOJFNBIPFOU-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 538081
Affinity DataIC50: 100nMAssay Description:Inhibition of PARP-1 enzymatic activities was measured using an HT Universal Colorimetric PARP Assay Kit (Trevigen, catalogue #4677-096-K) following ...More data for this Ligand-Target Pair