BDBM538070 4-(4-fluoro-3-(1-(3,5- difluoropyridin-2-yl)-4- oxido-1,4-azaphosphinan-4- yl)benzyl)phthalazin-1(2H)- one::US11248013, Example 28
SMILES Fc1cnc(N2CCP(=O)(CC2)c2cc(Cc3n[nH]c(=O)c4ccccc34)ccc2F)c(F)c1
InChI Key InChIKey=ZHSPDLMSKOGJLI-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 538070
Affinity DataIC50: 100nMAssay Description:Inhibition of PARP-1 enzymatic activities was measured using an HT Universal Colorimetric PARP Assay Kit (Trevigen, catalogue #4677-096-K) following ...More data for this Ligand-Target Pair