BDBM536491 (S)-5-(1-(2-((3-chloro- 2-fluoro-6-(3-methyl- morpholino)pyridin-4- yl)amino)-2-oxoethyl)- 4-oxo-4,6,7,8-tetra- hydro-1H-dipyrrolo [1,2-a:2',3'-d]pyrimi- din-3-yl)-2- hydroxy-3,4-dimethoxy- benzamide::US11242351, Compound I-70
SMILES COc1c(O)c(cc(-c2cn(CC(=O)Nc3cc(nc(F)c3Cl)N3CCOC[C@@H]3C)c3nc4CCCn4c(=O)c23)c1OC)C(N)=O
InChI Key InChIKey=WQVJGAYZYMTBON-UHFFFAOYSA-N
Data 1 Kd
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 536491
TargetB-cell lymphoma 6 protein [1-129]/Nuclear receptor corepressor 2 [1414-1429](Human)
Ontario Institute For Cancer Research (Oicr)
US Patent
Ontario Institute For Cancer Research (Oicr)
US Patent
Affinity DataKd: 255nMAssay Description:This assay was used to determine whether compounds inhibit the interaction between the BTB domain of BCL6 and a peptide derived from the BCL6 binding...More data for this Ligand-Target Pair