BDBM526517 US11186566, Compound 56

SMILES CC1(C)CN(c2nc(ccc2C(=O)NS(=O)(=O)c2ccccc2)-n2ccc(OCC3(CC3)C(F)(F)F)n2)C(C)(C)C1

InChI Key InChIKey=XYENWMOSXPHBOT-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 526517   

TargetCystic fibrosis transmembrane conductance regulator [1-507,509-1480](Human)
Vertex Pharmaceuticals

US Patent

LigandBDBM526517(US11186566, Compound 56)Copy SMILESCopy InChI

Affinity DataEC50:  550nMAssay Description:The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
4/9/2022
Entry Details
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