BDBM526515 US11186566, Compound 54

SMILES COc1ccc(cc1)S(=O)(=O)NC(=O)c1ccc(nc1N1C[C@@H](C)CC1(C)C)-n1ccc(OCC2(CC2)C(F)(F)F)n1

InChI Key InChIKey=ZDLUKUPLYJQBFK-UHFFFAOYSA-N

Data  1 EC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 526515   

TargetCystic fibrosis transmembrane conductance regulator [1-507,509-1480](Human)
Vertex Pharmaceuticals

US Patent

LigandBDBM526515(US11186566, Compound 54)Copy SMILESCopy InChI

Affinity DataEC50: <100nMAssay Description:The assay utilizes fluorescent voltage sensing dyes to measure changes in membrane potential using a fluorescent plate reader (e.g., FLIPR III, Molec...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
4/9/2022
Entry Details
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