BDBM518731 US11117865, Compound ZL0590

SMILES FC(F)(F)c1ccc(NC(=O)Nc2ccc(cc2)S(=O)(=O)N2CCC[C@@H]2CN2CCOCC2)cc1

InChI Key InChIKey=ZPMULUKHFNMJPF-UHFFFAOYSA-N

Data  18 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 18 hits for monomerid = 518731   

TargetBromodomain-containing protein 2 [91-163](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 824nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
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Ligand InfoPC cidPC sidSimilars

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TargetBromodomain-containing protein 4 [342-460](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 1.05E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

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TargetBromodomain-containing protein 4 [49-170](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 93nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

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TargetCREB-binding protein(Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+4nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

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TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 1.86E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetBromodomain testis-specific protein [22-138](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 2.35E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetBromodomain-containing protein 3 [326-398](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 2.01E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetBromodomain-containing protein 3 [51-123](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 2.27E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
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TargetBromodomain-containing protein 2 [364-436](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 1.28E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
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TargetBromodomain-containing protein 2 [91-163](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 824nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetBromodomain-containing protein 4 [342-460](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 1.05E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetBromodomain-containing protein 4 [49-170](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 93nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetCREB-binding protein(Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 1.00E+4nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetBromodomain testis-specific protein [287-359](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 1.86E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

Copy reaction URL

TargetBromodomain testis-specific protein [22-138](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 2.35E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetBromodomain-containing protein 3 [326-398](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 2.01E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetBromodomain-containing protein 3 [51-123](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 2.27E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

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TargetBromodomain-containing protein 2 [364-436](Human)
University Of Texas

US Patent

LigandBDBM518731(US11117865, Compound ZL0590)Copy SMILESCopy InChI

Affinity DataIC50: 1.28E+3nMAssay Description:Determine the binding ability of BRD4 compounds to bromodomains of BRD2 and BRD4. 96 well plate based commercial TR-FRET Assay kits (Cayman Chemical,...More data for this Ligand-Target Pair

Target InfoPDB
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In DepthDetails
Copy BDB DOIUS Patent

Copy reaction URL