BDBM511301 3-cyclopropyl-N-methyl-1-(7-(1-methyl-1H-pyrazol-4-yl)-6-(trifluoromethoxy)quinolin-4-yl)-5,6-dihydroimidazo[1,5-a]pyrazine-7(8H)-carboxamide::US11058688, Example 2
SMILES CNC(=O)N1CCn2c(C1)c(nc2C1CC1)-c1ccnc2cc(-c3cnn(C)c3)c(OC(F)(F)F)cc12
InChI Key InChIKey=IKYXDQOSZTUCJY-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 511301
Affinity DataIC50: 3nMAssay Description:5 nM GST-CBP(1081-1197) and 20 nM biotin-H4(1-21) Ac-K5/8/12/16 (AnaSpec. 64989) were incubated with varying concentrations of CBP inhibitors in 15 &...More data for this Ligand-Target Pair
Affinity DataIC50: 8.90E+3nMAssay Description:The binding of 2.5 nM of BRD4(49-170) to 10 nM biotin-H4(1-21) Ac-K5/8/12/16 (AnaSpec. 64989) was assessed following the same procedure described for...More data for this Ligand-Target Pair