BDBM50619059 CHEMBL5401978

SMILES OC(=O)Cc1cc(Cl)cc(OCCC2(CCN(CC2)c2nc3ccc(cc3s2)C(F)(F)F)N2CCCC2=O)c1

InChI Key InChIKey=KPGLBWBXEOAJKF-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50619059   

LigandPNGBDBM50619059(CHEMBL5401978)
Affinity DataEC50:  150nMAssay Description:Agonist activity at human PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed
LigandPNGBDBM50619059(CHEMBL5401978)
Affinity DataEC50:  410nMAssay Description:Agonist activity at mouse PPARdelta (138 to 441 residues) expressed in CHO-K1 cells co-transfected with GAL4 and pGluc reporter gene plasmid assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2024
Entry Details
PubMed