BDBM50602415 CHEMBL5190568

SMILES Cc1ccc(cc1)S(=O)(=O)Nc1cc(ccc1C)C(=O)NCc1ccc(C)nc1

InChI Key InChIKey=ZKRBQBKMMRYJKN-UHFFFAOYSA-N

Data  3 IC50

PDB links: 1 PDB ID matches this monomer.

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50602415   

TargetPotassium voltage-gated channel subfamily H member 2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50602415(CHEMBL5190568)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of hERG expressed in CHO cells by whole cell patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetSodium channel protein type 5 subunit alpha(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50602415(CHEMBL5190568)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Nav1.5 expressed in CHO cells by manual patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetVoltage-dependent L-type calcium channel subunit beta-2(Human)
Peking Union Medical College

Curated by ChEMBL
LigandPNGBDBM50602415(CHEMBL5190568)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human alpha1c/beta2a/alpha2delta1 Cav1.2 expressed in HEK293 cells assessed as effect on calcium flux by FLIPR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed