BDBM50596597 CHEMBL5182853

SMILES CCn1c2CCN(C)C(=O)c2cc1-c1ccncc1

InChI Key InChIKey=XRRPSTKWKIHULC-UHFFFAOYSA-N

Data  1 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50596597   

TargetSerine/threonine-protein kinase N2(Human)
University of Sussex

Curated by ChEMBL
LigandPNGBDBM50596597(CHEMBL5182853)
Affinity DataIC50: 350nMAssay Description:Inhibition of PKN2 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase N1(Human)
University of Sussex

Curated by ChEMBL
LigandPNGBDBM50596597(CHEMBL5182853)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase N2(Human)
University of Sussex

Curated by ChEMBL
LigandPNGBDBM50596597(CHEMBL5182853)
Affinity DataKi:  170nMAssay Description:Inhibition of PKN2 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed