BDBM50596595 CHEMBL5187643

SMILES CC(C)n1c2CCNC(=O)c2cc1-c1ccncc1

InChI Key InChIKey=MUKIIGVLQHTSFA-UHFFFAOYSA-N

Data  2 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50596595   

TargetSerine/threonine-protein kinase N2(Human)
University of Sussex

Curated by ChEMBL
LigandPNGBDBM50596595(CHEMBL5187643)
Affinity DataIC50: 140nMAssay Description:Inhibition of PKN2 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase N1(Human)
University of Sussex

Curated by ChEMBL
LigandPNGBDBM50596595(CHEMBL5187643)
Affinity DataIC50: 1.84E+3nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase N2(Human)
University of Sussex

Curated by ChEMBL
LigandPNGBDBM50596595(CHEMBL5187643)
Affinity DataKi:  70nMAssay Description:Inhibition of PKN2 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
TargetSerine/threonine-protein kinase N1(Human)
University of Sussex

Curated by ChEMBL
LigandPNGBDBM50596595(CHEMBL5187643)
Affinity DataKi:  920nMAssay Description:Inhibition of PKN1 (unknown origin) by TR-FRET-based tracer displacement assay dependent Cheng-Prusoff equation analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed