BDBM50596500 CHEMBL5180073

SMILES Cc1ccc(CC(O)=O)cc1OCCC1CCN(CC1)c1nc2ccc(Cl)cc2s1

InChI Key InChIKey=WWMKSYGAMJOHCB-UHFFFAOYSA-N

Data  10 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 10 hits for monomerid = 50596500   

LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  637nMAssay Description:Transactivation of Gal4-fused human PPARalpha expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  542nMAssay Description:Transactivation of Gal4-fused human PPARgamma expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  16nMAssay Description:Transactivation of Gal4-fused human PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  71nMAssay Description:Transactivation of Gal4-fused mouse PPARdelta expressed in CHO cells co expressing pG5-Luc reporterMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/22/2023
Entry Details
PubMed
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  16nMAssay Description:Agonist activity at Gal4-fused human PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  637nMAssay Description:Agonist activity at Gal4-fused human PPAR-alpha ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  542nMAssay Description:Agonist activity at Gal4-fused human PPAR-gamma ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  71nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-delta ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  1.13E+3nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-alpha ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed
LigandPNGBDBM50596500(CHEMBL5180073)
Affinity DataEC50:  744nMAssay Description:Agonist activity at Gal4-fused mouse PPAR-gamma ligand binding domain expressed in CHO-K1 cells assessed as receptor transactivation incubated for 24...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2024
Entry Details
PubMed