BDBM50596334 CHEMBL5205647
SMILES NC(=S)c1ccc(cc1)C(=O)NC1CCN(Cc2ccccc2)CC1
InChI Key InChIKey=MDRXXGMJEJFONZ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50596334
TargetPotassium voltage-gated channel subfamily H member 2(Human)
University of Catania
Curated by ChEMBL
University of Catania
Curated by ChEMBL
Affinity DataIC50: 6.80E+3nMAssay Description:Inhibition of human ERG potassium channel expressed in CHO-K1 cells by Qube-automated patch clamp assayMore data for this Ligand-Target Pair
Affinity DataKi: 94nMAssay Description:Displacement of [3H]-(+)-pentazocine from Dunkin-Hartley guinea pig brain cortex Sigma 1 receptor incubated for 150 mins by liquid scintillation coun...More data for this Ligand-Target Pair
Affinity DataKi: 1.13E+3nMAssay Description:Displacement of [3H]-DTG from Sprague-Dawley rat liver Sigma 2 receptor incubated for 120 mins in presence of [3H]-(+)-pentazocine by liquid scintill...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-DAMGO from Sprague-Dawley rat brain membrane mu opioid receptor incubated for 45 mins by liquid scintillation counting analysisMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-(2-D-Ala)[Tyrosy1-3,5-]-DELTORPHIN II from Sprague-Dawley rat brain membrane delta opioid receptor incubated for 45 mins by liqu...More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]-U69593 from Dunkin-Hartley guinea pig brain membrane kappa opioid receptor incubated for 30 mins by liquid scintillation countin...More data for this Ligand-Target Pair