BDBM50593188 CHEMBL5205658

SMILES CCc1ccccc1COc1ccc(cc1)C1C2=C(CC(C)(C)CC2=O)OC2=C1C(=O)CC(C)(C)C2

InChI Key InChIKey=PXKQLLRQPSFAPI-UHFFFAOYSA-N

Data  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50593188   

TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593188(CHEMBL5205658)
Affinity DataEC50:  2.34E+7nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced ERK1/2 phosphorylation level by measuring Leu-enkephal...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed
TargetDelta-type opioid receptor(Human)
Monash University (Parkville Campus)

Curated by ChEMBL
LigandPNGBDBM50593188(CHEMBL5205658)
Affinity DataEC50:  1.62E+8nMAssay Description:Inhibition of human DOR expressed in CHO cells assessed as reduction in Leu-enkephalin induced cAMP level by measuring Leu-enkephalin pEC50 measured ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/20/2023
Entry Details
PubMed