BDBM50582145 CHEMBL5084070

SMILES Oc1ccc(cc1)-c1ccc2c(n[nH]c2c1)-c1ccc(cc1)N1CCN(CCN2CCOC2=O)CC1

InChI Key InChIKey=PCSUKDRXNKOZEL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50582145   

TargetFibroblast growth factor receptor 2(Human)
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50582145(CHEMBL5084070)
Affinity DataIC50: 9.60E+4nMAssay Description:Inhibition of wild type FGFR2 (unknown origin) (461 to 763 residues) transfected in Escherichia coli BL21(DE3) cells using Tyr04 peptide as substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed
TargetFibroblast growth factor receptor 1(Human)
University of Leeds

Curated by ChEMBL
LigandPNGBDBM50582145(CHEMBL5084070)
Affinity DataIC50: 449nMAssay Description:Inhibition of FGFR1 (unknown origin) (458 to 765 residues) transfected in Escherichia coli BL21(DE3) cells using Tyr04 peptide as substrate incubated...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/5/2023
Entry Details Article
PubMed