BDBM50581734 CHEMBL5081182

SMILES CN(C)c1noc(n1)-c1cccc(CNc2ccc3[nH]nc(C(O)=O)c3c2)c1O

InChI Key InChIKey=QZFNTDYKERMDQJ-UHFFFAOYSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50581734   

Target2-Hydroxyacid oxidase 1(Human)
X-Chem

Curated by ChEMBL
LigandPNGBDBM50581734(CHEMBL5081182)
Affinity DataIC50: 37nMAssay Description:Inhibition of human recombinant HAO1 assessed as detecting hydrogen peroxide using glycolic acid as substrate preincubated for 30 min followed by sub...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-Hydroxyacid oxidase 1(Human)
X-Chem

Curated by ChEMBL
LigandPNGBDBM50581734(CHEMBL5081182)
Affinity DataIC50: 1.30E+4nMAssay Description:Inhibition of human recombinant HAO1 assessed as fluorescent intensity using hydrogen peroxide as substrate by HRP interference detection assayMore data for this Ligand-Target Pair
In DepthDetails Article
PubMed
Target2-Hydroxyacid oxidase 1(Human)
X-Chem

Curated by ChEMBL
LigandPNGBDBM50581734(CHEMBL5081182)
Affinity DataEC50:  1.70E+4nMAssay Description:Inhibition of human recombinant HAO1 expressed in CHO cells co-transformed with a vector expressing glycolate oxidase assessed as cell rescue from CH...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed