BDBM50579191 CHEMBL4869006

SMILES CC(C)Oc1ccc(cc1)-c1cc(Nc2ccnc3cc(ccc23)-c2ccc(cc2)S(C)(=O)=O)ccn1

InChI Key InChIKey=CDPNFJNZLHNIHC-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50579191   

TargetTGF-beta receptor type-1(Human)
University of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50579191(CHEMBL4869006)
Affinity DataIC50: 127nMAssay Description:Inhibition of human TGFbeta receptor 1 in human HEK293 cells preincubated for 24 hrs followed by addition of TGFbeta1 and measured after 24 hrs by lu...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed