BDBM50572927 CHEMBL4862024

SMILES CCOc1ccc(cc1C(F)(F)F)C1=NNC(=O)O[C@H]1C

InChI Key InChIKey=GKCRJVINJPUMCL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50572927   

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50572927(CHEMBL4862024)
Affinity DataIC50: 6nMAssay Description:Inhibition of human full length PDE3A expressed in Sf9 cells measured after 60 mins by [3H]-cAMP Scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3B(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50572927(CHEMBL4862024)
Affinity DataIC50: 7nMAssay Description:Inhibition of human full length PDE3B expressed in Sf9 cells measured after 60 mins by [3H]-cAMP Scintillation proximity assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2022
Entry Details Article
PubMed