BDBM50564378 CHEMBL4787157

SMILES COc1cc(\C=C2\C(=N)N3N=C(SC3=NC2=O)C(F)(F)F)ccc1O

InChI Key InChIKey=CQYCTLSWCZSZBJ-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50564378   

TargetSRSF protein kinase 1(Human)
University of Trento

Curated by ChEMBL
LigandPNGBDBM50564378(CHEMBL4787157)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of recombinant human SRPK1 expressed in Escherichia coli using RS peptide as substrate incubated for 15 mins in presence of ATP by Kinase-...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetSRSF protein kinase 1(Human)
University of Trento

Curated by ChEMBL
LigandPNGBDBM50564378(CHEMBL4787157)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of SRPK1 (unknown origin) using SRSF1 Arg-Ser (RS) peptide (NH2-RSPSYGRSRSRSRSRSRSRSRSNSRSRSY-OH) as substrate incubated for 10 mins in pr...More data for this Ligand-Target Pair
In DepthDetails
PubMed
TargetSRSF protein kinase 2(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50564378(CHEMBL4787157)
Affinity DataIC50: 203nMAssay Description:Inhibition of SRPK2 (unknown origin) incubated for 10 mins in presence of ATP by Kinase-Glo assayMore data for this Ligand-Target Pair
In DepthDetails
PubMed