BDBM50559597 CHEMBL4776935

SMILES COc1cc(F)c2nc(N3CC[C@@H](F)[C@H](N)C3)n(Cc3ncc(Cl)cn3)c2c1

InChI Key InChIKey=LAVRDVHZGGEPJZ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50559597   

TargetShort transient receptor potential channel 6(Human)
Smith, Gambrell & Russell

Curated by ChEMBL
LigandPNGBDBM50559597(CHEMBL4776935)
Affinity DataIC50: 0.400nMAssay Description:Inhibition of human TRPC6 channel transfected in HEK293 cells assessed as intracellular calcium level by FLIPR assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed