BDBM50559507 CHEMBL4764314

SMILES Oc1cc(cc(O)c1-c1cc(F)cc(F)c1)C(=O)c1ccccc1

InChI Key InChIKey=BILQKQJGNQPIPM-UHFFFAOYSA-N

Data  2 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50559507   

TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559507(CHEMBL4764314)
Affinity DataEC50:  1.70E+3nMAssay Description:Inverse agonist activity at human recombinant cannabinoid CB2 receptor expressed in HEK cells transfected with CNG assessed as increase in cAMP level...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559507(CHEMBL4764314)
Affinity DataEC50:  8.91E+3nMAssay Description:Inverse agonist activity at cannabinoid CB2 receptor in human U2OS cells assessed as induction of beta-arrestin recruitment using CCF4/AM as substrat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 1(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559507(CHEMBL4764314)
Affinity DataKi:  1.08E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB1 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetCannabinoid receptor 2(Human)
University of Tennessee Health Science Center

Curated by ChEMBL
LigandPNGBDBM50559507(CHEMBL4764314)
Affinity DataKi:  1.63E+3nMAssay Description:Displacement of [3H]-CP55940 from human recombinant cannabinoid CB2 receptor expressed in HEK cell membranes incubated for 1.5 hrs by liquid scintill...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed