BDBM50552415 CHEMBL4749601
SMILES NC(=O)[C@H](N([C@@H]1CCc2c1cc(Cl)cc2F)C(=O)c1ccccc1)c1ccccc1
InChI Key InChIKey=ZLDDOCXDTRTKDS-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50552415
TargetTransient receptor potential cation channel subfamily M member 8(Human)
Kissei Pharmaceutical
Curated by ChEMBL
Kissei Pharmaceutical
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Antagonist activity at human TRPM8 transfected in HEK293T cells assessed as reduction in menthol-induced calcium influx measured after 60 mins by Flu...More data for this Ligand-Target Pair
Affinity DataEC50: 4.70E+3nMAssay Description:Activation of human PXR ligand binding domain incubated for 1 hr by TR-FRET assayMore data for this Ligand-Target Pair