BDBM50552410 CHEMBL4795385

SMILES NC(=O)[C@H](N([C@@H]1CCc2c1cc(Cl)cc2F)C(=O)c1cccnc1N)c1ccccc1

InChI Key InChIKey=UQWXSZBNADPSOU-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50552410   

TargetTransient receptor potential cation channel subfamily M member 8(Human)
Kissei Pharmaceutical

Curated by ChEMBL

LigandBDBM50552410(CHEMBL4795385)Copy SMILESCopy InChI

Affinity DataIC50: 170nMAssay Description:Antagonist activity at human TRPM8 transfected in HEK293T cells assessed as reduction in menthol-induced calcium influx measured after 60 mins by Flu...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
3/24/2022
Entry Details Article
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