BDBM50547930 CHEMBL4782190

SMILES COc1cc(OC(F)(F)F)ccc1Oc1cc(OC)c(c(F)c1C(=O)Nc1ccnc(c1)C(N)=O)C(F)(F)F

InChI Key InChIKey=FTGXJMQFAMEXKW-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50547930   

TargetSodium channel protein type 10 subunit alpha(Human)
Temple University

Curated by ChEMBL
LigandPNGBDBM50547930(CHEMBL4782190)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human Nav1.8 expressed in HEK cells applied electrical stimulus 10 Hz for 10 seconds measuring relaxation to the resting state followed...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed