BDBM50529947 CHEMBL4461175

SMILES Cc1ccc(CNC(=O)[C@@H]2COCCCCCCOc3ccccc3C(=O)N[C@@H](CC(=O)NCC(C)(C)C)C(=O)N2)cc1

InChI Key InChIKey=JYIINRSQFLSIQL-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50529947   

TargetProteasome subunit beta type-5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50529947(CHEMBL4461175)
Affinity DataIC50: 67nMAssay Description:Inhibition of human hepatic cell derived 20s constitutive proteasome beta5 chymotrypsin-like activity using Suc-WLA-AMC as substrate preincubated for...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-5(Human)
Zhejiang University

Curated by ChEMBL
LigandPNGBDBM50529947(CHEMBL4461175)
Affinity DataIC50: 67nMAssay Description:Inhibition of human hepatic cell derived 20s constitutive proteasome beta5 chymotrypsin-like activity using Suc-WLA-AMC as substrate preincubated for...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed