BDBM50521875 CHEMBL4464323

SMILES Cc1ccc2nc3N(CCn3c2c1)C(=O)Cc1nc2nc(C)cc(C)n2n1

InChI Key InChIKey=SQFKHNCTIWBRQW-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50521875   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50521875(CHEMBL4464323)Copy SMILESCopy InChI

Affinity DataIC50: 416nMAssay Description:Inhibition of human PDE10A using cAMP as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by HTRF detecti...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/23/2021
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