BDBM50521873 CHEMBL4469276

SMILES Cc1cc(C)n2nc(CC(=O)N3CCn4c3nc3ccccc43)nc2n1

InChI Key InChIKey=UDBWOTVGWIHJNG-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50521873   

TargetcAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A(Human)
Astellas Pharma

Curated by ChEMBL

LigandBDBM50521873(CHEMBL4469276)Copy SMILESCopy InChI

Affinity DataIC50: 52nMAssay Description:Inhibition of human PDE10A using cAMP as substrate preincubated for 30 mins followed by substrate addition and measured after 60 mins by HTRF detecti...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

In Depth
Date in BDB:
2/23/2021
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