BDBM50520466 CHEMBL4564309
SMILES CCOc1ccc(CN2CCCC2)cc1CNC(=O)[C@@H](N)Cc1c(C)cc(O)cc1C
InChI Key InChIKey=DYFWFMUVZWQKQN-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50520466
Affinity DataEC50: 168nMAssay Description:Agonist activity at human MOR expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by by liquid scin...More data for this Ligand-Target Pair
Affinity DataEC50: >6.00E+3nMAssay Description:Agonist activity at human KOR expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by by liquid scin...More data for this Ligand-Target Pair
Affinity DataEC50: 1.36E+3nMAssay Description:Agonist activity at human DOR expressed in CHO cell membranes assessed as stimulation of [35S]-GTPgammaS binding incubated for 1 hr by by liquid scin...More data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Displacement of [3H]diprenorphine from human MOR expressed in CHO cell membranes incubated for 1 hr by liquid scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Displacement of [3H]diprenorphine from human DOR expressed in CHO cell membranes incubated for 1 hr by liquid scintillation counting assayMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Displacement of [3H]diprenorphine from human KOR expressed in CHO cell membranes incubated for 1 hr by liquid scintillation counting assayMore data for this Ligand-Target Pair