BDBM50511108 CHEMBL4558185
SMILES [H][C@]12N(CCC[C@@]1(CC)C=C(C(=O)OC)n1c2c(CCNC(=O)c2ccc(Br)cc2)c2ccccc12)C#N
InChI Key InChIKey=IUXSPRUXYTWDEG-UHFFFAOYSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50511108
Affinity DataIC50: 5.20E+3nMAssay Description:Antagonist activity at human CCR8 expressed in CHOK1 cells assessed as reduction in CCL1-induced beta-arrestin 2 recruitment incubated for 30 mins fo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:Antagonist activity at human Gi/o-coupled FPR1 expressed in CHOK1 cells assessed as reduction in WKYMVm-NH2-induced beta-arrestin 2 recruitment incub...More data for this Ligand-Target Pair
Affinity DataIC50: 5.77E+3nMAssay Description:Antagonist activity at human Gq-coupled NPSR1b expressed in human U2OS cells assessed as inhibition in neuropeptide S-induced beta-arrestin 2 recruit...More data for this Ligand-Target Pair
Affinity DataIC50: 2.43E+3nMAssay Description:Antagonist activity at human Gq-coupled PRLHR expressed in CHOK1 cells assessed as inhibition in prolactin releasing peptide (1 to 31)-induced beta-a...More data for this Ligand-Target Pair