BDBM50502326 CHEMBL4460217

SMILES COc1ncc(cc1NS(C)(=O)=O)-c1ccc2ncnc(NCCN3CCCCC3)c2c1

InChI Key InChIKey=GKGFBPSWYYWNMK-UHFFFAOYSA-N

Data  1 IC50

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50502326   

TargetPhosphatidylinositol 4,5-bisphosphate 3-kinase catalytic subunit alpha isoform(Human)
Xi'An Jiaotong University

Curated by ChEMBL

LigandBDBM50502326(CHEMBL4460217)Copy SMILESCopy InChI

Affinity DataIC50: 12nMAssay Description:Inhibition of PI3K alpha (unknown origin) using lipid substrate measured after 40 mins in presence of ATP by Kinase-Glo plus reagent based luminescen...More data for this Ligand-Target Pair

Target InfoPDBKEGG
UniProtKB/SwissProt
GoogleScholar

Ligand InfoPC cidPC sidSimilars

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