BDBM50470536 CHEMBL4292798

SMILES [H][C@]1([C@@H](C)CC)[C@@H](OC1=O)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](C(C)C)C(=O)NCc1ccccc1

InChI Key InChIKey=FXAMLICIOFJBJL-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50470536   

TargetmRNA cap guanine-N7 methyltransferase(Human)
New Mexico Institute of Mining and Technology

Curated by ChEMBL
LigandPNGBDBM50470536(CHEMBL4292798)
Affinity DataIC50: 2.92E+3nMAssay Description:Inhibition of yeast 20S proteasome beta2 subunit using SUC-RLR-AMC as substrate pretreated for 30 mins followed by substrate addition and measured af...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetProteasome subunit beta type-5(Human)
New Mexico Institute of Mining and Technology

Curated by ChEMBL
LigandPNGBDBM50470536(CHEMBL4292798)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of 20S proteasome beta5 subunit in human Jurkat cell lysate using Suc-LLVY-AMC as substrate pretreated for 30 mins followed by substrate a...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetmRNA cap guanine-N7 methyltransferase(Human)
New Mexico Institute of Mining and Technology

Curated by ChEMBL
LigandPNGBDBM50470536(CHEMBL4292798)
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of yeast 20S proteasome beta1 subunit using fluorescent substrate pretreated for 30 mins followed by substrate addition and measured after...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed