BDBM50469986 CHEMBL313149::US11542274, Compound 039

SMILES O=C1Cc2cc(ccc2N1)-c1ccncc1

InChI Key InChIKey=OQWVVJNJCRCQSJ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50469986   

TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Human)
Sterling Winthrop Pharmaceuticals Research Division

Curated by ChEMBL
LigandPNGBDBM50469986(CHEMBL313149 | US11542274, Compound 039)
Affinity DataIC50: 5.30E+3nMAssay Description:In vitro inhibitory activity against cAMP phosphodiesterase III in dog aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetProtein cereblon(Human)
Agency For Science, Technology and Research (A*Star)

US Patent
LigandPNGBDBM50469986(CHEMBL313149 | US11542274, Compound 039)
Affinity DataIC50: 2.00E+5nMAssay Description:Fluorescence quenching end point measurements were performed in black polystyrene 384-plates on Tecan Safire monochromator reader with the following ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2023
Entry Details
Go to US Patent