BDBM50469422 CHEMBL4293167

SMILES C\N=C(\NCCCC[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)[C@H](Cc1ccccc1)NC(=O)CNC(=O)CN)C(=O)N[C@@H](Cc1ccccc1)C(N)=O)N(C)C

InChI Key InChIKey=DTNIJMWZXRUYPC-UHFFFAOYSA-N

Data  1 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50469422   

TargetPyroglutamylated RF-amide peptide receptor(Human)
Normandy University

Curated by ChEMBL
LigandPNGBDBM50469422(CHEMBL4293167)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed
TargetPyroglutamylated RF-amide peptide receptor(Human)
Normandy University

Curated by ChEMBL
LigandPNGBDBM50469422(CHEMBL4293167)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as increase Ca2+ mobilization after 3 mins by Fluo-4 AM-based ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2020
Entry Details Article
PubMed