BDBM50468283 CHEMBL4278563
SMILES CCCC[C@H](NC(=O)[C@@H](Cc1ccccc1)NC(=O)[C@H](Cc1cnc[nH]1)NC(C)=O)C(=O)N[C@@H](Cc1c[nH]c2ccccc12)C(N)=O
InChI Key InChIKey=XVOPWUWRTVGXCT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 8 hits for monomerid = 50468283
Affinity DataIC50: 1.00E+3nMAssay Description:Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 928nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells after 3 mins by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 120nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells after 3 mins by cAMP assayMore data for this Ligand-Target Pair
Affinity DataEC50: 52nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells after 3 mins by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting analysisMore data for this Ligand-Target Pair
Affinity DataEC50: 37nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells after 3 mins by cAMP assayMore data for this Ligand-Target Pair
Affinity DataIC50: 65nMAssay Description:Displacement of [125I]-[Nle4,d-Phe7]-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting analysisMore data for this Ligand-Target Pair