BDBM50463963 CHEBI:85252::CHEMBL1482206

SMILES CC\C=C/C\C=C/C\C=C/C\C=C/C\C=C/C\C=C/CCC(=O)NCCO

InChI Key InChIKey=GEEHOLRSGZPBSM-UHFFFAOYSA-N

Data  4 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50463963   

TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM50463963(CHEBI:85252 | CHEMBL1482206)
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
National Research Council (Cnr)

Curated by ChEMBL
LigandPNGBDBM50463963(CHEBI:85252 | CHEMBL1482206)
Affinity DataIC50: 1.63E+3nMAssay Description:Antagonist activity at recombinant rat TRPV2 expressed in HEK293 cells assessed as inhibition of CBD-induced Ca2+ levels preincubated for 5 mins foll...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Ehime University

Curated by ChEMBL
LigandPNGBDBM50463963(CHEBI:85252 | CHEMBL1482206)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human FAAH expressed in baculovirus infected Sf9 cells using N-(6-methoxypyridin-3-yl)octanamide as substrate measured for 15 mins by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetFatty-acid amide hydrolase 1(Human)
Ehime University

Curated by ChEMBL
LigandPNGBDBM50463963(CHEBI:85252 | CHEMBL1482206)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human FAAH expressed in baculovirus infected Sf9 cells using N-(6-methoxypyridin-3-yl)octanamide as substrate measured for 15 mins by f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed