BDBM50459019 CHEMBL4207505

SMILES FC(F)(F)Oc1cccc(Cl)c1-c1ccc2NC(=O)Cc2c1

InChI Key InChIKey=KDQVOHZGLRUPLF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50459019   

TargetGlutamate receptor 1/Voltage-dependent calcium channel gamma-8 subunit(Human)
Janssen Research & Development

Curated by ChEMBL
LigandPNGBDBM50459019(CHEMBL4207505)
Affinity DataIC50: 16nMAssay Description:Modulation of recombinant human GluA1 flop isoform/TARPgamma8 expressed in HEK293F cells assessed as blockade of glutamate-induced calcium flux by ca...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed