BDBM50456974 CHEMBL3621636

SMILES Nc1nc(\C=C\CNC(=O)c2cc(Br)c[nH]2)c[nH]1

InChI Key InChIKey=KHJREOQCERRAME-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50456974   

TargetPotassium voltage-gated channel subfamily A member 1(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Kv1.1 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 3(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human Kv1.3 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 5(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of human Kv1.5 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 6(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human Kv1.6 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 4(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human Kv1.4 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily A member 2(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50456974(CHEMBL3621636)
Affinity DataIC50: 3.00E+4nMAssay Description:Inhibition of human Kv1.2 expressed in CHO cells at -80 mV holding potential by whole cell automated patch clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed