BDBM50455150 CHEMBL4207102

SMILES Fc1ccc(cc1)[C@H]1NCCO[C@@H]1OCc1cc(F)c(cc1F)S(=O)(=O)Nc1ncns1

InChI Key InChIKey=RXTKDBFVUHSEEI-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50455150   

TargetSodium channel protein type 9 subunit alpha(Human)
Bristol-Myers Squibb Research and Development

Curated by ChEMBL
LigandPNGBDBM50455150(CHEMBL4207102)
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at recombinant human Nav1.7 expressed in HEK293 cells assessed as reduction in channel current at -60 mV holding potential after ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed